Found 361 recordings
DICL IDIon ChannelCompound FunctionSpeciesValueReferences
DICL_CP_0307400Gamma-aminobutyric acid receptor subunit alpha-1AntagonistRattus norvegicus (Rat)Ki: 6600 nM10.1016/S0014-2999(97)89183-2, 9226416
DICL_CP_0307539Gamma-aminobutyric acid receptor subunit alpha-1AntagonistRattus norvegicus (Rat)IC50: >10000 nM10.1016/S0014-2999(97)89183-2, 9226416
DICL_CP_0309761Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2AgonistRattus norvegicus (Rat)EC50: 50000 (GABA-mimetic action) nM10.1021/jm010903i, 11606122
DICL_CP_0309762Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2AgonistRattus norvegicus (Rat)EC50: 4100 (GABA-modulatory action) nM10.1021/jm010903i, 11606122
DICL_CP_0310030Gamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2AntagonistRattus norvegicus (Rat)Ki: 0.8 nM10.1021/jm00052a019, 7799410
DICL_CP_0311017Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2Allosteric ModulatorRattus norvegicus (Rat)EC50: 44000 nM10.1021/acs.jmedchem.8b00859, 30289721
DICL_CP_0311018Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2Allosteric ModulatorRattus norvegicus (Rat)EC50: 41000 nM10.1021/acs.jmedchem.8b00859, 30289721
DICL_CP_0313005Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2 (beta-3/N265 mutation)Allosteric ModulatorRattus norvegicus (Rat)EC50: 103000 nM10.1021/acs.jmedchem.8b00859, 30289721
DICL_CP_0313006Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2 (beta-3/F289S mutation)Allosteric ModulatorRattus norvegicus (Rat)EC50: 171000 nM10.1021/acs.jmedchem.8b00859, 30289721
DICL_CP_0313007Gamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2Allosteric ModulatorRattus norvegicus (Rat)EC50: 13000 nM10.1021/acs.jmedchem.8b00859, 30289721
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